Something interesting about 3066-84-0

Compounds in my other articles are similar to this one(8-Bromoguanine)Recommanded Product: 3066-84-0, you can compare them to see their pros and cons in some ways,such as convenient, effective and so on.

In organic chemistry, atoms other than carbon and hydrogen are generally referred to as heteroatoms. The most common heteroatoms are nitrogen, oxygen and sulfur. Now I present to you an article called Synthesis of 6- and 8-alkynylated purines and their ribonucleosides by the coupling of halopurines with alkynes, published in 1982, which mentions a compound: 3066-84-0, mainly applied to alkynylated purine; nucleotide alkynylated purine; alkynylation purine; coupling halopurine alkyne; cytokinin activity alkynylated purine, Recommanded Product: 3066-84-0.

Coupling reactions of 6-iodo- or 6-chloropurine with alkynes in the presence of (PPh3)2PdCl2-CuI catalyst in Et3N to give 6-alkynylated purines was achieved by the use of dipolar aprotic solvent as cosolvent. Under the reaction conditions, ribonucleoside as well as its tri-O-acetate of 6-chloropurine also gave the corresponding alkynylated products in high yields. Though similar reaction for 8-bromo derivatives of adenineand guanine gave poor yields, the 8-alkynylated free bases could be obtained by acid hydrolysis of the alkynylated ribonucleosides. 6-Alkynylated purines exhibited moderate to weak cytokinin activity in Amaranthus test.

Compounds in my other articles are similar to this one(8-Bromoguanine)Recommanded Product: 3066-84-0, you can compare them to see their pros and cons in some ways,such as convenient, effective and so on.

Reference:
Tetrahydrofuran – Wikipedia,
Tetrahydrofuran | (CH2)3CH2O – PubChem