Brief introduction of 5061-21-2

5061-21-2 2-Bromo-4-butanolide 95463, aTetrahydrofurans compound, is more and more widely used in various fields.

5061-21-2, 2-Bromo-4-butanolide is a Tetrahydrofurans compound, ?involved in a variety of chemical synthesis. Rlated chemical reaction is continuously updated

5061-21-2, (Step 1) To a solution of 2-amino-5-nitrophenol (2.00 g, 13 mmol) in DMF (20 mL) were added 3-bromo-dihydrofuran-2-one and potassium carbonate (2.1 g, 15.57 mmol), and the mixture was stirred at 80C for 4 hr under nitrogen atmosphere. The reaction mixture was allowed to be cooled to room temperature, and filtered through Celite, and the filtrate was concentrated under reduced pressure. The obtained residue was dissolved in ethyl acetate, and the solution was washed with water and saturated brine, and dried over sodium sulfate, and the solvent was evaporated under reduced pressure. The obtained yellow solid was washed with pentane to give 2-(2-hydroxyethyl)-7-nitro-4H-benzo[1,4]oxazin-3-one (2.5 g, 80.9%) as a yellow solid. MS (API) :239 (M+H)

5061-21-2 2-Bromo-4-butanolide 95463, aTetrahydrofurans compound, is more and more widely used in various fields.

Reference£º
Patent; Takeda Pharmaceutical Company Limited; YAMAMOTO, Satoshi; SHIRAI, Junya; FUKASE, Yoshiyuki; SATO, Ayumu; KOUNO, Mitsunori; TOMATA, Yoshihide; OCHIDA, Atsuko; YONEMORI, Kazuko; ODA, Tsuneo; IMADA, Takashi; YUKAWA, Tomoya; (238 pag.)EP2975031; (2016); A1;,
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